SCHEMBL20003172

SCHEMBL20003172

CC(Oc1ccccc1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA4 P22748 1/20 0.40
PDK1 Q15118 3/20 0.38
PDK2 Q15119 3/20 0.38
PDK3 Q15120 3/20 0.38
PDK4 Q16654 3/20 0.38
TSHR P16473 2/20 0.38
LTA4H P09960 2/20 0.38
MAPK1 P28482 1/20 0.36
PPARA Q07869 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
PPARG P37231 2/20 0.35
ALDH1A1 P00352 2/20 0.35
RIPK1 Q13546 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9770338 0.80 CA4 (0.43) CA4PDK1PDK2PDK3PDK4
SCHEMBL10477060 0.80 CA4 (0.43) CA4PDK1PDK2PDK3PDK4
SCHEMBL20002025 0.79 CA1 (0.50) CA4PDK1PDK2PDK3PDK4
SCHEMBL20002023 0.79 GAA (0.40) PPARAMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL16886265 0.77 CA4 (0.37) CA4PDK1PDK2PDK3PDK4
SCHEMBL7481516 0.77 PDK1 (0.39) CA4PDK1PDK2PDK3PDK4
SCHEMBL13039942 0.76 CA4 (0.40) CA4PDK1PDK2PDK3PDK4
SCHEMBL821312 0.76 CA4 (0.40) CA4PDK1PDK2PDK3PDK4
SCHEMBL24615573 0.75 LTA4H (0.41) CA4PDK1PDK2PDK3PDK4
SCHEMBL6000951 0.75 LTA4H (0.41) CA4PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed