SCHEMBL20002023

SCHEMBL20002023

CC(Oc1ccc(F)cc1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
NFE2L2 Q16236 1/20 0.38
CASR P41180 1/20 0.35
RORC P51449 4/20 0.35
ACHE P22303 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
PPARA Q07869 1/20 0.34
HSD11B1 P28845 2/20 0.34
GPR3 P46089 1/20 0.34
CNR1 P21554 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002025 0.82 CA1 (0.50) GAANFE2L2ACHECYP3A4MAPT
SCHEMBL19477799 0.81 GAA (0.42) GAANFE2L2CASRRORCACHE
SCHEMBL20003172 0.79 CA4 (0.40) RORCCYP1A2CYP2D6CYP2C19MEN1
SCHEMBL16886216 0.78 GAA (0.38) GAANFE2L2CASRRORCACHE
SCHEMBL4977051 0.78 NFE2L2 (0.41) GAANFE2L2CASRACHECYP1A2
SCHEMBL10603546 0.76 GAA (0.42) GAANFE2L2RORCACHEMAPT
SCHEMBL255560 0.75 GPR3 (0.52) GAACASRMAPTHSD11B1GPR3
SCHEMBL3160868 0.74 NFE2L2 (0.39) GAANFE2L2CASRACHECYP1A2
SCHEMBL22967387 0.73 HSPB1 (0.48) GAANFE2L2MEN1MAPTKMT2A
SCHEMBL10641834 0.73 GAA (0.40) GAANFE2L2RORCMAPTHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed