SCHEMBL20002327

SCHEMBL20002327

N#Cc1ccc(SC2CCN(C(=O)N3CCC(C(=O)O)CC3)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
NOTUM Q6P988 1/20 0.41
AKR1C3 P42330 1/20 0.41
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
EPHX2 P34913 1/20 0.38
HSD11B1 P28845 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
POLB P06746 3/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 1/20 0.36
PDK2 Q15119 1/20 0.35
RORC P51449 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PAX8 Q06710 1/20 0.34
GPR119 Q8TDV5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21824778 0.85 MAOA (0.51) MAOAMAOBDDB1CRBNEPHX2
SCHEMBL21825012 0.85 MAOA (0.51) MAOAMAOBDDB1CRBNEPHX2
SCHEMBL20002297 0.84 NOTUM (0.47) NOTUMAKR1C3HSD11B1ITGB3ITGA2B
SCHEMBL20003024 0.77 NOTUM (0.44) NOTUMAKR1C3EPHX2HSD11B1KMT2A
SCHEMBL24117778 0.76 GPR119 (0.56) MAOAMAOBKMT2AMAPTALDH1A1
SCHEMBL21824803 0.76 GPR119 (0.56) MAOAMAOBKMT2AMAPTALDH1A1
SCHEMBL21887032 0.76 GPR119 (0.56) MAOAMAOBKMT2AMAPTALDH1A1
SCHEMBL21887036 0.71 MAOA (0.57) MAOAMAOBDDB1CRBNRAB9A
SCHEMBL20002879 0.70 NPC1 (0.44) KMT2AL3MBTL1RAB9AALDH1A1
SCHEMBL7962518 0.69 NAMPT (0.57) MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed