SCHEMBL20002297

SCHEMBL20002297

O=C(O)C1CCN(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.47
AKR1C3 P42330 1/20 0.43
HSD11B1 P28845 3/20 0.41
RORC P51449 3/20 0.40
CCR5 P51681 1/20 0.39
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
MGLL Q99685 1/20 0.38
KMT2A Q03164 1/20 0.38
RAB9A P51151 2/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
NPC1 O15118 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003024 0.92 NOTUM (0.44) NOTUMAKR1C3HSD11B1CCR5MAPT
SCHEMBL20002879 0.86 NPC1 (0.44) CCR5L3MBTL1KMT2ARAB9AGRIN1
SCHEMBL20002936 0.85 CCR5 (0.46) AKR1C3HSD11B1CCR5MAPTKMT2A
SCHEMBL20002407 0.85 SMN1; SMN2 (0.41) AKR1C3CCR5KMT2ARAB9AGRIN1
SCHEMBL20002327 0.84 MAOA (0.45) NOTUMAKR1C3HSD11B1RORCMAPT
SCHEMBL20002612 0.82 RORC (0.36) NOTUMRORCCCR5KMT2ARAB9A
SCHEMBL20002294 0.81 PTPN11 (0.36) RORCCCR5KMT2AGRIN1GRIN2B
SCHEMBL20002972 0.81 L3MBTL1 (0.41) NOTUMHSD11B1RORCMAPTL3MBTL1
SCHEMBL20003026 0.79 RORC (0.47) NOTUMHSD11B1RORCCCR5MAPT
SCHEMBL20002255 0.79 CCR5 (0.49) HSD11B1RORCCCR5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed