SCHEMBL20002582

SCHEMBL20002582

[O-][S+](c1ccc(F)cc1)C1CCN(Cc2ccccc2)C1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.56
BACE1 P56817 7/20 0.56
BCHE P06276 6/20 0.56
DRD4 P21917 2/20 0.46
DRD2 P14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002873 1.00 ACHE (0.56) ACHEBACE1BCHEDRD4DRD2
SCHEMBL20002589 0.83 BCHE (0.43) ACHEBACE1BCHEDRD4
SCHEMBL20003099 0.83 BCHE (0.43) ACHEBACE1BCHE
SCHEMBL7023032 0.76 HTR2A (0.49) ACHE
SCHEMBL2729881 0.74 DRD4 (0.48) DRD4
SCHEMBL7027090 0.74 HTR2A (0.52)
SCHEMBL6041781 0.73 SLC18A3 (0.58) ACHEBACE1BCHE
SCHEMBL20002470 0.72 PDE4B (0.31) ACHEBACE1BCHE
SCHEMBL19493714 0.72 SLC18A3 (0.70) ACHEBACE1BCHEDRD4
SCHEMBL8553491 0.71 ACHE (0.57) ACHEBACE1BCHEDRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed