SCHEMBL20002589

SCHEMBL20002589

Cc1cc([S+]([O-])C2CCN(Cc3ccccc3)C2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BCHE P06276 12/20 0.43
ACHE P22303 12/20 0.43
BACE1 P56817 11/20 0.43
DRD4 P21917 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
SCN4A P35499 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003099 0.91 BCHE (0.43) BCHEACHEBACE1SCN4A
SCHEMBL20002582 0.83 ACHE (0.56) BCHEACHEBACE1DRD4
SCHEMBL20002873 0.83 ACHE (0.56) BCHEACHEBACE1DRD4
SCHEMBL2729881 0.73 DRD4 (0.48) DRD4SIGMAR1
SCHEMBL20003010 0.70 RORC (0.43)
SCHEMBL20002976 0.69 RORC (0.43) DRD4
SCHEMBL2345413 0.68 MAOA (0.59) ACHE
SCHEMBL1552524 0.68 DRD4 (0.59) DRD4SIGMAR1
SCHEMBL13186450 0.67 ACHE (0.52) BCHEACHEBACE1SIGMAR1
SCHEMBL27573515 0.67 LTA4H (0.51) BCHEACHEBACE1DRD4TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed