SCHEMBL20002470

SCHEMBL20002470

O=CN1CCC([S+]([O-])c2ccc(F)cc2)C1

nearest known ligand 0.31

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.31
TACR1 P25103 1/20 0.31
NOTUM Q6P988 1/20 0.31
TSHR P16473 1/20 0.31
PKM P14618 1/20 0.30
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
BACE1 P56817 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002854 0.83 RORC (0.42) TSHRPKM
SCHEMBL20002664 0.82 TSHR (0.41) TSHRPKMNPC1RAB9AATM
SCHEMBL20002631 0.74 HSD11B1 (0.33) NOTUMPKMNPC1RAB9AATM
SCHEMBL20002873 0.72 ACHE (0.56) BCHEACHEBACE1
SCHEMBL20002582 0.72 ACHE (0.56) BCHEACHEBACE1
SCHEMBL20002698 0.70 HSD11B1 (0.47) TSHR
SCHEMBL20002706 0.70 HSD11B1 (0.47) TSHR
SCHEMBL29051099 0.70 RAB9A (0.49) PDE4BTACR1NPC1RAB9AATM
SCHEMBL29051117 0.70 RAB9A (0.49) PDE4BTACR1NPC1RAB9AATM
SCHEMBL29051096 0.70 RAB9A (0.49) PDE4BTACR1NPC1RAB9AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed