SCHEMBL20003607

SCHEMBL20003607

COc1cc(NC(=O)C2(C(N)=O)CC2)ccc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 9/20 0.56
GRM4 Q14833 2/20 0.49
FLT1 P17948 2/20 0.47
AURKB Q96GD4 2/20 0.47
RAB9A P51151 1/20 0.46
AXL P30530 4/20 0.46
KDR P35968 2/20 0.46
EGFR P00533 2/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.44
MERTK Q12866 2/20 0.43
AURKA O14965 1/20 0.43
RIPK2 O43353 1/20 0.43
ABCB11 O95342 1/20 0.43
ABL1 P00519 1/20 0.43
ERBB2 P04626 1/20 0.43
NTRK1 P04629 1/20 0.43
LCK P06239 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18256946 0.85 MET (0.54) METGRM4FLT1AURKBAXL
SCHEMBL18256970 0.85 MET (0.52) METGRM4FLT1AURKBRAB9A
SCHEMBL22210776 0.84 MET (0.53) METGRM4FLT1AURKBAXL
SCHEMBL18256945 0.84 MET (0.53) METGRM4FLT1AURKBAXL
SCHEMBL20003906 0.83 KDR (0.56) METRAB9AKDRRETKIT
SCHEMBL28524761 0.77 NPC1 (0.54) RAB9AKMT2A
SCHEMBL22643534 0.77 MET (0.47) METGRM4FLT1AURKBAXL
SCHEMBL30616270 0.76 ALDH1A1 (0.45) METFLT1AURKBRAB9AAXL
SCHEMBL16136597 0.76 MET (0.67) METFLT1AURKBAXLKDR
SCHEMBL27778083 0.76 KDR (0.43) METRAB9AKDRKMT2AABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299369-A1 PYRIDO-AZAHETERECYDIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2018-03-28 EP disclosed