SCHEMBL20003906

SCHEMBL20003906

NC(=O)C1(C(=O)Nc2ccc(F)c(F)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.56
EPHB4 P54760 2/20 0.56
TEK Q02763 2/20 0.56
MET P08581 11/20 0.51
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
RET P07949 1/20 0.43
KIT P10721 1/20 0.43
PDGFRA P16234 1/20 0.43
FLT3 P36888 1/20 0.43
NAMPT P43490 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30074424 0.90 KDR (0.57) KDREPHB4TEKMETNPC1
SCHEMBL453535 0.87 RAB9A (0.53) KDREPHB4TEKMETNPC1
SCHEMBL20003607 0.83 MET (0.56) KDRTEKMETRAB9ARET
SCHEMBL18256911 0.83 KDR (0.52) KDREPHB4TEKMETNPC1
SCHEMBL407809 0.82 ALDH1A1 (0.56) KDRMETSMN1; SMN2RETKIT
Hydrochloric Acid SCHEMBL29453838 0.81 ALDH1A1 (0.55) KDRMETSMN1; SMN2RETKIT
Water SCHEMBL2458178 0.81 ALDH1A1 (0.55) KDRMETSMN1; SMN2RETKIT
SCHEMBL27778083 0.80 KDR (0.43) KDREPHB4TEKMETNPC1
SCHEMBL28520615 0.80 MEN1 (0.53) METNPC1RAB9A
SCHEMBL22210779 0.80 KDR (0.49) KDREPHB4TEKMETNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105153028-B Compound as c-Met kinase inhibitor 南京爱德程医药科技有限公司 2019-03-26 CN claimed
CN-112142619-B 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2023-01-10 CN disclosed
CN-112142619-A 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2020-12-29 CN disclosed
EP-3299369-A1 PYRIDO-AZAHETERECYDIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2018-03-28 EP disclosed