SCHEMBL20004451

SCHEMBL20004451

Ic1ccc(COCc2ccncc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.50
IDO1 P14902 2/20 0.50
HDAC8 Q9BY41 1/20 0.50
APP P05067 12/20 0.48
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
TSHR P16473 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL508682 0.86 CYP3A4 (0.64) CYP3A4IDO1APPHRH4HRH3
SCHEMBL492258 0.86 TSHR (0.52) CYP3A4TSHRLOXL2
Hydrochloric Acid SCHEMBL27794104 0.84 TSHR (0.50) CYP3A4TSHRLOXL2
SCHEMBL3541962 0.79 HDAC8 (0.57) CYP3A4HDAC8TSHRLOXL2
SCHEMBL1825953 0.79 APP (0.73) HDAC8APP
SCHEMBL20004502 0.78 KCNH2 (0.52) CYP3A4IDO1TSHRLOXL2
SCHEMBL14156900 0.78 IDO1 (0.50) IDO1
SCHEMBL22537715 0.78 RAB9A (0.46) CYP3A4TSHRLOXL2
SCHEMBL14156909 0.78 IDO1 (0.50) CYP3A4IDO1APP
SCHEMBL3500426 0.77 TSHR (0.71) CYP3A4IDO1APPTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018055316-A1 COMPOUNDS FOR USING IN IMAGING AND PARTICULARLY FOR THE DIAGNOSIS OF NEURODEGENERATIVE DISEASES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-29 WO disclosed