SCHEMBL20004950

SCHEMBL20004950

CN(C)CCOc1cccc2c1C(C)(C)c1[nH]c3c(c1C2=O)CCC(N)=C3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.38
NOS1 P29475 4/20 0.38
NOS2 P35228 4/20 0.38
HTR7 P34969 3/20 0.35
ALK Q9UM73 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ESR1 P03372 1/20 0.33
HTR1B P28222 1/20 0.33
PDE5A O76074 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE7A Q13946 1/20 0.32
PDE1C Q14123 1/20 0.32
TIPARP Q7Z3E1 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21766971 0.76 ALK (0.50) ALK
SCHEMBL29962304 0.70 ALK (0.69) ALK
SCHEMBL898103 0.70 ALK (0.69) ALK
SCHEMBL17154500 0.66 HTR7 (0.51) HTR7KDM4EALDH1A1SMN1; SMN2HTR1B
SCHEMBL7791992 0.66 HTR7 (0.54) HTR7KDM4EALDH1A1SMN1; SMN2HTR1B
SCHEMBL898280 0.65 ALK (0.68) ALK
SCHEMBL29962592 0.65 ALK (0.68) ALK
SCHEMBL3583265 0.64 ADORA2A (0.49) NOS3NOS1NOS2HTR7KDM4E
Hydrochloric Acid SCHEMBL11606266 0.64 KCNA3 (0.61) HTR7KDM4EALDH1A1SMN1; SMN2HTR1B
SCHEMBL21443318 0.62 HTR7 (0.37) NOS3NOS1NOS2HTR7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed