SCHEMBL20006909

SCHEMBL20006909

O=C(Nc1cc(Cl)cc(NC(=O)c2ccc(-c3cccc(-c4cccc(-c5ccc(C(=O)Oc6cc(Cl)cc(OC(=O)c7ccc(-c8ccccc8)nc7)c6)cn5)c4)c3)nc2)c1)c1ccc(-c2ccccc2)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
BAZ2B Q9UIF8 1/20 0.45
P4HTM Q9NXG6 1/20 0.44
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
KMT2A Q03164 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
MEN1 O00255 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGDS O60760 1/20 0.42
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
LDHA P00338 1/20 0.41
MCHR1 Q99705 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19933546 0.85 LDHA (0.55) BAZ2BHPGDSLDHA
SCHEMBL19933523 0.85 TRPV1 (0.60) TRPV1SIRT2SIRT1SIRT3BAZ2B
SCHEMBL18573404 0.80 TRPV1 (0.49) TRPV1SIRT2SIRT1SIRT3BAZ2B
SCHEMBL18573397 0.79 BAZ2B (0.68) TRPV1SIRT2SIRT1SIRT3BAZ2B
SCHEMBL18573164 0.79 LDHA (0.63) TRPV1BAZ2BP4HTMHPGDSNPC1
SCHEMBL22059853 0.78 LDHA (0.47) BAZ2BHPGDSLDHA
SCHEMBL22563324 0.78 TRPV1 (0.53) TRPV1SIRT2SIRT1SIRT3BAZ2B
SCHEMBL23018779 0.78 TRPV1 (0.55) TRPV1SIRT2SIRT1SIRT3BAZ2B
SCHEMBL21125569 0.76 LDHA (0.49) BAZ2BHPGDSNPC1ALDH1A1RAB9A
SCHEMBL23018724 0.76 HPGDS (0.53) TRPV1SIRT2SIRT1SIRT3BAZ2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069196-A1 BINUCLEAR METAL COMPLEXES AND ELECTRONIC DEVICES, IN PARTICULAR ORGANIC ELECTROLUMINESCENT DEVICES CONTAINING SAID METAL COMPLEXES MERCK PATENT GMBH (DE) 2018-04-19 WO disclosed
WO-2018054798-A1 BINUCLEAR METAL COMPLEXES FOR USE AS EMITTERS IN ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2018-03-29 WO disclosed