SCHEMBL20008488

SCHEMBL20008488

C=CCCN(CC)c1cc(-c2cccnc2)cnc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP2A6 P11509 7/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP2E1 P05181 2/20 0.38
CYP2B6 P20813 2/20 0.38
GRM5 P41594 1/20 0.35
CYP2D6 P10635 1/20 0.35
PDGFRB P09619 2/20 0.35
PDGFRA P16234 2/20 0.35
FYN P06241 1/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
EGFR P00533 1/20 0.34
GBA1 P04062 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008358 0.77 VRK1 (0.31)
SCHEMBL18136476 0.68 CYP2A6 (0.56) CYP19A1CYP11B1CYP11B2CYP2A6CYP3A4
SCHEMBL20008162 0.66 CRHR1 (0.35)
SCHEMBL14934101 0.65 CYP2A6 (0.56) CYP19A1CYP11B1CYP11B2CYP2A6CYP3A4
SCHEMBL12072374 0.64 CHRNB2 (0.41) CYP3A4CYP2C9CYP2C19CYP2B6ALDH1A1
SCHEMBL18134393 0.63 CYP2A6 (0.48) CYP19A1CYP11B1CYP11B2CYP2A6CYP3A4
SCHEMBL20008535 0.62 VRK1 (0.31)
SCHEMBL29078028 0.61 PDGFRB (0.56) CYP19A1CYP11B1CYP11B2CYP2A6CYP3A4
SCHEMBL12024774 0.61 PDE2A (0.49)
SCHEMBL23812543 0.61 CYP11B1 (0.50) CYP19A1CYP11B1CYP11B2CYP2A6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed