SCHEMBL20009265

SCHEMBL20009265

C=C(Nc1cnc(C)c(C(=N)/C=C\C)c1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 9/20 0.45
BRAF P15056 5/20 0.43
CYP2C9 P11712 2/20 0.43
LCK P06239 7/20 0.42
MAPK14 Q16539 3/20 0.42
KDR P35968 1/20 0.42
CSF1R P07333 2/20 0.41
JAK2 O60674 1/20 0.41
PDGFRB P09619 1/20 0.41
FGFR1 P11362 1/20 0.41
EPHB4 P54760 1/20 0.41
PTK2 Q05397 1/20 0.41
KCNQ3 O43525 2/20 0.40
KCNQ2 O43526 2/20 0.40
KCNE1 P15382 2/20 0.40
KCNQ1 P51787 2/20 0.40
KCNQ5 Q9NR82 1/20 0.40
BLK P51451 2/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20009576 0.74 RAF1 (0.40) BRAFRAF1
SCHEMBL20008505 0.69 RAF1 (0.47) BRAFRAF1
SCHEMBL19623099 0.69 LMNA (0.68)
SCHEMBL4434874 0.66 KCNQ3 (0.65) BTKBRAFLCKMAPK14KDR
SCHEMBL16036513 0.66 KCNQ3 (0.65) BTKBRAFCYP2C9LCKMAPK14
SCHEMBL24275085 0.66 KCNQ3 (0.65) BTKBRAFCYP2C9LCKMAPK14
SCHEMBL20009609 0.65 BTK (0.32) BTKBRAFCYP2C9
SCHEMBL21877180 0.65 KCNQ3 (0.63) BTKBRAFCYP2C9LCKMAPK14
SCHEMBL26075509 0.65 KCNQ3 (0.63) BTKBRAFCYP2C9LCKMAPK14
SCHEMBL19073411 0.64 BRAF (0.53) BRAFLCKMAPK14KDRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed