SCHEMBL20009309

SCHEMBL20009309

C/C=C\C(=N/CC)c1cc(NC(=O)c2ccnc(C(C)(C)F)c2)cnc1C

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 19/20 0.47
BRAF P15056 13/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25996456 0.71 RAF1 (0.44) RAF1BRAF
SCHEMBL17591679 0.69 RAF1 (0.56) RAF1BRAF
SCHEMBL29427240 0.69 RAF1 (0.56) RAF1BRAF
SCHEMBL25984339 0.68 RAF1 (0.70) RAF1BRAF
SCHEMBL25985505 0.67 RAF1 (0.59) RAF1BRAF
SCHEMBL19355675 0.66 RAF1 (0.46) RAF1BRAF
SCHEMBL25984092 0.66 LMNA (0.56) RAF1BRAF
SCHEMBL21297359 0.66 RAF1 (0.50) RAF1BRAF
SCHEMBL20008346 0.66 BRAF (0.86) RAF1BRAF
SCHEMBL25984369 0.65 RAF1 (0.60) RAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed