SCHEMBL29427240

SCHEMBL29427240

Cc1ncc(NC(=O)c2ccnc(C(F)(F)F)c2)cc1Br

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 15/20 0.56
BRAF P15056 14/20 0.56
NPC1 O15118 1/20 0.52
LMNA P02545 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17591679 1.00 RAF1 (0.56) RAF1BRAFNPC1LMNARAB9A
SCHEMBL30405369 0.84 NPC1 (0.56) RAF1BRAFNPC1LMNARAB9A
SCHEMBL23482203 0.84 NPC1 (0.56) RAF1BRAFNPC1LMNARAB9A
SCHEMBL16036520 0.84 RAF1 (0.59) RAF1BRAF
SCHEMBL26165531 0.84 SLC6A3 (0.47) NPC1LMNARAB9ASMN1; SMN2
SCHEMBL16036513 0.83 KCNQ3 (0.65) RAF1BRAFLMNARAB9A
SCHEMBL30016396 0.81 LMNA (0.51) RAF1BRAFNPC1LMNARAB9A
SCHEMBL28637538 0.81 LMNA (0.51) RAF1BRAFNPC1LMNARAB9A
SCHEMBL17542187 0.80 LMNA (0.59) NPC1LMNARAB9ASMN1; SMN2
SCHEMBL25984181 0.79 RAF1 (0.63) RAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116761801-A Heterocyclic compounds having protein kinase inhibitory activity, pharmaceutical compositions containing the same, and methods of preparing and using the same 四川科伦博泰生物医药股份有限公司 2023-09-15 CN disclosed
EP-3962484-A1 INHIBITORS OF RAF KINASES Kinnate Biopharma Inc. (US) 2022-03-09 EP disclosed