SCHEMBL20011291

SCHEMBL20011291

C=C1NC(=O)c2c(ncn2C)N1C

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.31
CYP3A4 P08684 2/20 0.30
PMP22 Q01453 2/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30
BLM P54132 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10039865 0.71 PIK3CD (0.30) GDA
SCHEMBL11987584 0.71 ALDH1A1 (0.32) GDAALDH1A1TSHR
SCHEMBL2136936 0.67 GDA (0.32) GDACYP3A4PMP22ALDH1A1LMNA
SCHEMBL20011085 0.67 GDA (0.32) GDACYP3A4PMP22ALDH1A1LMNA
SCHEMBL19090554 0.62 HCAR3 (0.31)
SCHEMBL19090548 0.62 BRD4 (0.39) ALDH1A1TSHR
SCHEMBL9910655 0.61 GDA (0.33) GDACYP3A4PMP22ALDH1A1LMNA
SCHEMBL10104855 0.60 GDA (0.32) GDACYP3A4PMP22ALDH1A1LMNA
SCHEMBL15624085 0.60
SCHEMBL31685444 0.58 ALDH1A1 (0.38) GDAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299371-A1 HYDROXYL PURINE COMPOUNDS AND USE THEREOF GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2018-03-28 EP disclosed