SCHEMBL20021142

SCHEMBL20021142

Cc1cc2nc(C3N=CC=CC3C)ccc2c(-c2ccc(Cl)cc2)c1[C@H](OC(C)(C)C)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.42
CYP3A4 P08684 2/20 0.41
KDM4E B2RXH2 1/20 0.31
DHODH Q02127 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245283 0.83 PSIP1 (0.49) PSIP1CYP3A4
SCHEMBL243700 0.82 PSIP1 (0.50) PSIP1CYP3A4KDM4EDHODH
SCHEMBL244914 0.81 PSIP1 (0.51) PSIP1CYP3A4KDM4EDHODH
SCHEMBL244717 0.81 PSIP1 (0.51) PSIP1CYP3A4KDM4EDHODH
SCHEMBL3304151 0.79 PSIP1 (0.48) PSIP1CYP3A4KDM4EDHODH
SCHEMBL3312489 0.79 PSIP1 (0.44) PSIP1CYP3A4
SCHEMBL244312 0.79 PSIP1 (0.49) PSIP1CYP3A4KDM4EDHODH
SCHEMBL243122 0.79 PSIP1 (0.49) PSIP1CYP3A4KDM4EDHODH
SCHEMBL20021147 0.79 PSIP1 (0.49) PSIP1CYP3A4KDM4EDHODH
SCHEMBL243123 0.79 PSIP1 (0.49) PSIP1CYP3A4KDM4EDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed