SCHEMBL20021157

SCHEMBL20021157

Cc1cc2nc(NCc3ccncc3)ccc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.39
PTGDR2 Q9Y5Y4 3/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
CLK4 Q9HAZ1 2/20 0.37
ALDH1A1 P00352 2/20 0.36
POLB P06746 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021122 0.86 KDM4E (0.52) KDM4EMEN1KMT2ASMN1; SMN2PTGDR2
SCHEMBL3324004 0.82 KDM4E (0.48) KDM4ESMN1; SMN2PTGDR2ALDH1A1MAPT
SCHEMBL20020801 0.80 KDM4E (0.46) KDM4ESMN1; SMN2PTGDR2
SCHEMBL3297610 0.79 KDM4E (0.54) KDM4EMEN1KMT2ASMN1; SMN2PTGDR2
SCHEMBL246129 0.79 PSIP1 (0.42) KDM4EMEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL3303954 0.78 KDM4E (0.53) KDM4EMEN1KMT2ASMN1; SMN2PTGDR2
SCHEMBL15182622 0.78 MEN1 (0.38) KDM4EMEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL20020750 0.78 KDM4E (0.41) KDM4EMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL3326729 0.77 ACHE (0.47) KDM4EMEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL3323941 0.77 KDM4E (0.51) KDM4EMEN1KMT2ASMN1; SMN2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed