SCHEMBL2002122

SCHEMBL2002122

COc1ccc2c(c1)c(C(=O)c1nnc(-c3cccnc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C19 P33261 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 2/20 0.41
MEN1 O00255 1/20 0.41
RGS12 O14924 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
GNAI1 P63096 1/20 0.41
PMP22 Q01453 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
PLA2G2A P14555 3/20 0.41
KDM4E B2RXH2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004592 0.93 ALOX5AP (0.41) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2004532 0.92 PTGES2 (0.42) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2002253 0.91 PLA2G2A (0.46) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2C9
SCHEMBL2004484 0.91 KDM4E (0.38) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2C9
SCHEMBL2008741 0.91 PTGES2 (0.44) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2002430 0.91 MAPK1 (0.46) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2C9
SCHEMBL1999749 0.90 ALOX5AP (0.43) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2003185 0.90 PTGES2 (0.41) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2001738 0.90 CYP3A4 (0.44) PTGES2CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2008862 0.89 PLA2G2A (0.49) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed