SCHEMBL2008741

SCHEMBL2008741

Cc1ccc2c(c1)c(C(=O)c1nnc(-c3cccnc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 5/20 0.44
FAAH O00519 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 3/20 0.39
NPC1 O15118 3/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RECQL P46063 1/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004532 0.94 PTGES2 (0.42) PTGES2FAAHCYP1A2CYP3A4CYP2D6
SCHEMBL2003185 0.91 PTGES2 (0.41) PTGES2FAAHCYP1A2CYP3A4CYP2D6
SCHEMBL2011368 0.91 PTGES2 (0.41) PTGES2FAAHKDM4EALDH1A1MAPT
SCHEMBL2005825 0.91 RET (0.38) PTGES2FAAHRAB9ANPC1KDM4E
SCHEMBL2002122 0.91 PTGES2 (0.41) PTGES2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2006683 0.90 MAPK1 (0.47) PTGES2FAAHCYP1A2CYP3A4CYP2C9
SCHEMBL2000862 0.90 PTGES2 (0.43) PTGES2FAAHCYP1A2CYP3A4CYP2D6
SCHEMBL2003594 0.90 FAAH (0.47) PTGES2FAAHCYP1A2CYP3A4CYP2D6
SCHEMBL2009227 0.90 CYP1A2 (0.42) PTGES2FAAHCYP1A2CYP3A4CYP2D6
SCHEMBL2007848 0.89 PTGES2 (0.45) PTGES2FAAHKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed