SCHEMBL20030832

SCHEMBL20030832

CCOC(=O)Cc1c(C)cc2nc(-c3ccc4c(c3)c(N3CCN(C)CC3)nn4C)sc2c1-c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HRH4 Q9H3N8 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPK10 P53779 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
FPR1 P21462 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HDAC3 O15379 1/20 0.33
MTOR P42345 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17547135 0.91 KDM4E (0.35) KDM4EHRH4HPGDALDH1A1HTT
SCHEMBL20030918 0.88 KDM4E (0.39) KDM4ETDP1L3MBTL1SMN1; SMN2HPGD
SCHEMBL20030761 0.87 KDM4E (0.36) KDM4ETDP1L3MBTL1SMN1; SMN2HPGD
SCHEMBL20030973 0.86 KDM4E (0.43) KDM4ETDP1L3MBTL1SMN1; SMN2HPGD
SCHEMBL19906245 0.85 HDAC3 (0.37) KDM4EHRH4ALDH1A1MEN1KMT2A
SCHEMBL20030976 0.84 SMN1; SMN2 (0.35) KDM4ETDP1L3MBTL1SMN1; SMN2HPGD
SCHEMBL20030828 0.84 BRD4 (0.34) KDM4EHRH4HPGDMEN1KMT2A
SCHEMBL31114867 0.84 BRD4 (0.34) KDM4EHRH4HPGDMEN1KMT2A
SCHEMBL19906008 0.84 TACR1 (0.36) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL20030670 0.83 L3MBTL1 (0.32) KDM4ETDP1L3MBTL1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064080-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING HIV INFECTION GILEAD SCIENCES, INC. (US) 2018-04-05 WO disclosed