SCHEMBL20031893

SCHEMBL20031893

CCOc1ccc2c(c1)CCc1c3c(c4c(c1-2)-c1ccc(OC)cc1CC4)C(=O)N(c1ccccc1)C3=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SLC11A2 P49281 1/20 0.45
MIF P14174 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAP3K9 P80192 3/20 0.42
MAP3K11 Q16584 3/20 0.42
CYP24A1 Q07973 2/20 0.42
CYP27A1 Q02318 1/20 0.42
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25016974 0.92 ALDH1A1 (0.52) GAAALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL22703031 0.86 ESR1 (0.50) GAAALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL20031637 0.81 BRD4 (0.42) GAAALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL25017625 0.80 BRD4 (0.50)
SCHEMBL25016866 0.78 ITGB3 (0.40) ACHE
SCHEMBL25016973 0.77 CYP1A2 (0.46) ALDH1A1KDM4ECYP1A2SLC11A2MIF
SCHEMBL22703045 0.76 MGLL (0.37) GAAALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL25018113 0.75 BRD4 (0.45) ACHE
SCHEMBL25017621 0.74 ESR1 (0.56) KDM4EMIFNTRK1POLBMAPK14
SCHEMBL25017019 0.74 ITGB3 (0.38) GAAALDH1A1KDM4EL3MBTL1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed