SCHEMBL20031904

SCHEMBL20031904

CCCCCCOc1ccc2c(c1)CCc1c(C#N)c(C#N)c3c(c1-2)-c1ccc(OCCCCCC=O)cc1CC3

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRA P10827 2/20 0.43
THRB P10828 2/20 0.43
MAOB P27338 6/20 0.39
EGFR P00533 4/20 0.38
PTPN11 Q06124 2/20 0.36
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20031911 0.95 MAOB (0.41) THRATHRBMAOBEGFR
SCHEMBL22702989 0.92 THRA (0.47) THRATHRBMAOBEGFRPTPN11
SCHEMBL20031909 0.90 MAOB (0.43) MAOBEGFR
SCHEMBL20031873 0.90 MAOB (0.38) MAOBEGFR
SCHEMBL20031890 0.90 MAOB (0.38) MAOBEGFRALDH1A1MEN1KMT2A
SCHEMBL20031650 0.90 MAOB (0.38) THRATHRBMAOBEGFR
SCHEMBL22683257 0.89 MAOB (0.39) MAOBEGFRALDH1A1L3MBTL1MEN1
SCHEMBL22703070 0.87 THRA (0.35) THRATHRBMAOBEGFR
SCHEMBL22683261 0.85 MEN1 (0.46) THRATHRBMAOBEGFRPTPN11
SCHEMBL22683269 0.84 BRD4 (0.52) MAOBEGFRMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed