SCHEMBL20031922

SCHEMBL20031922

CC(C)c1ccc(Cl)cc1-c1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.41
AKR1C2 P52895 3/20 0.41
TRPV3 Q8NET8 1/20 0.38
F11 P03951 1/20 0.38
SCN9A Q15858 1/20 0.38
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
HTT P42858 1/20 0.37
KMO O15229 2/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NOTUM Q6P988 1/20 0.36
PDE2A O00408 1/20 0.36
CNR1 P21554 1/20 0.35
AR P10275 1/20 0.34
HSD11B1 P28845 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
PDE3B Q13370 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21507822 0.88 KDM4E (0.43) AKR1C3AKR1C2SCN9ANOTUMTMPRSS4
SCHEMBL21507816 0.87 F11 (0.38) AKR1C3AKR1C2F11SCN9ANOTUM
SCHEMBL18713986 0.85 AKR1C3 (0.42) AKR1C3AKR1C2TRPV3F11SCN9A
SCHEMBL21507998 0.81 PTGS2 (0.44) LMNATP53HTTTSHR
SCHEMBL20032372 0.80 AKR1C3 (0.39) AKR1C3AKR1C2TRPV3F11SCN9A
SCHEMBL16574088 0.80 SCN9A (0.48) AKR1C3AKR1C2SCN9AKMOCYP3A4
SCHEMBL21507823 0.77 TRPV1 (0.49) LMNATP53HTTCYP3A4
SCHEMBL21508375 0.77 AKR1C3 (0.43) AKR1C3AKR1C2LMNAHTTCYP3A4
SCHEMBL3017108 0.76 AKR1C3 (0.39) AKR1C3AKR1C2TRPV3SCN9AKMO
SCHEMBL4547920 0.76 GABRA1 (0.42) LMNATP53HTTCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018060949-A1 TRYPTOPHAN HYDROXYLASE INHIBITORS FOR USE IN THE TREATMENT OF LIVER DISEASES ROIVANT SCIENCES GMBH (CH) 2018-04-05 WO disclosed