SCHEMBL20033899

SCHEMBL20033899

CCOC(=O)c1c(C)cn2cc(-c3cccc(Cl)c3)nc2c1-c1cc(F)c2c(c1C)CCCO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.40
DGAT1 O75907 1/20 0.36
SOAT1 P35610 1/20 0.36
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX5 P09917 3/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
BCHE P06276 2/20 0.34
TP53 P04637 2/20 0.34
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CACNB4 O00305 1/20 0.33
CACNA1A O00555 1/20 0.33
CACNA1G O43497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17029033 0.93 NR1I2 (0.39) NR1I2DGAT1SOAT1GABRA2GABRB2
SCHEMBL17029006 0.93 NR1I2 (0.41) NR1I2L3MBTL1TP53MAPTPDE4B
SCHEMBL17029005 0.90 NR1I2 (0.42) NR1I2PDE4APDE4BPDE4CKDM4E
SCHEMBL20344833 0.90 NR1I2 (0.41) NR1I2PDE4APDE4BPDE4CKMT2A
SCHEMBL17039259 0.89 NR1I2 (0.39) NR1I2L3MBTL1TRPM8TP53MAPT
SCHEMBL17039244 0.88 NR1I2 (0.42) NR1I2GABRA2GABRB2L3MBTL1BCHE
SCHEMBL20344788 0.88 NR1I2 (0.42) NR1I2GABRA2GABRB2L3MBTL1BCHE
SCHEMBL20344789 0.86 NR1I2 (0.37) NR1I2MAPTKDM4EALDH1A1HPGD
SCHEMBL17039260 0.85 NR1I2 (0.50) NR1I2
SCHEMBL17029021 0.83 NR1I2 (0.45) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938271-B2 Inhibitors of human immunodeficiency virus replication VIIV Healthcare UK (No.5) Limited (GB) 2018-04-10 US disclosed