SCHEMBL20037056

SCHEMBL20037056

CC(=O)OCC(=O)Nc1c(C)nn(C)c1C

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.60
NR2F2 P24468 1/20 0.51
ALDH1A1 P00352 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TSHR P16473 3/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
KLK6 Q92876 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846945 0.78 GAA (0.70) GAANR2F2ALDH1A1L3MBTL1TSHR
SCHEMBL20037038 0.78 GAA (0.70) GAANR2F2ALDH1A1L3MBTL1TSHR
SCHEMBL20037138 0.76 LMNA (0.68) ALDH1A1LMNAHTTKLK6SMN1; SMN2
SCHEMBL20037047 0.76 KLK6 (0.74) ALDH1A1LMNAHTTKLK6SMN1; SMN2
SCHEMBL20037154 0.73 KLK6 (0.59) ALDH1A1LMNAHTTKLK6SMN1; SMN2
SCHEMBL20037114 0.72 KLK6 (0.55) ALDH1A1LMNAHTTKLK6SMN1; SMN2
SCHEMBL20037205 0.72 KLK6 (0.55) ALDH1A1LMNAHTTKLK6SMN1; SMN2
SCHEMBL20037102 0.72 NPC1 (0.59) GAAALDH1A1TSHRHSD17B10LMNA
SCHEMBL9223302 0.70 GAA (0.54) GAANR2F2ALDH1A1L3MBTL1TSHR
SCHEMBL4491737 0.69 USP2 (0.51) ALDH1A1L3MBTL1LMNASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed