SCHEMBL20037038

SCHEMBL20037038

Cc1nn(C)c(C)c1NC(=O)CO

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.70
TSHR P16473 3/20 0.54
ALDH1A1 P00352 3/20 0.54
HSD17B10 Q99714 1/20 0.54
LMNA P02545 2/20 0.50
HTT P42858 2/20 0.50
KDM4E B2RXH2 2/20 0.47
NR2F2 P24468 1/20 0.47
MAPT P10636 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.43
RIPK1 Q13546 1/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KLK6 Q92876 1/20 0.42
TP53 P04637 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846945 0.85 GAA (0.70) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL50204 0.79 GAA (0.61) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL20037056 0.78 GAA (0.60) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL12156243 0.74 GAA (0.56) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL12788582 0.74 GAA (0.56) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL9223302 0.73 GAA (0.54) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL20037309 0.73 LMNA (0.77) ALDH1A1LMNAHTTKDM4EMAPT
SCHEMBL20037281 0.73 ALDH1A1 (0.77) ALDH1A1LMNAHTTKDM4EMAPT
SCHEMBL10310296 0.69 GAA (0.50) GAATSHRALDH1A1HSD17B10LMNA
SCHEMBL6917528 0.69 GAA (0.48) GAATSHRALDH1A1HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed