SCHEMBL20037601

SCHEMBL20037601

Nc1ccc(N2C3CCC2CNC3)cn1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.49
CHRNA4 P43681 3/20 0.49
OPRM1 P35372 1/20 0.44
USP25 Q9UHP3 2/20 0.38
USP28 Q96RU2 1/20 0.38
PIM1 P11309 1/20 0.36
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20038082 0.80 OPRM1 (0.44) CHRNB2CHRNA4OPRM1USP25USP28
SCHEMBL17796315 0.80 MTOR (0.46) CHRNB2CHRNA4PIK3CAMTOR
SCHEMBL611573 0.79 OPRM1 (0.45) CHRNB2CHRNA4OPRM1PIK3CAMTOR
SCHEMBL23089115 0.79 CHRNB2 (0.44) CHRNB2CHRNA4PIK3CAMTORROCK2
SCHEMBL23089117 0.79 CHRNB2 (0.44) CHRNB2CHRNA4PIK3CAMTORROCK2
SCHEMBL23089116 0.79 CHRNB2 (0.44) CHRNB2CHRNA4PIK3CAMTORROCK2
SCHEMBL23215232 0.76 HTR2A (0.42) CHRNB2CHRNA4OPRM1CHRNB4CHRNA3
SCHEMBL20249258 0.76 OPRM1 (0.41) CHRNB2CHRNA4OPRM1USP25USP28
SCHEMBL18291649 0.76 OPRM1 (0.41) OPRM1USP25USP28ROCK2ROCK1
SCHEMBL31111805 0.76 MAPK14 (0.39) CHRNB2CHRNA4OPRM1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed