SCHEMBL20040871

SCHEMBL20040871

O=CNc1ccc2c(c1)C(F)(F)CCO2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.41
KDR P35968 1/20 0.41
MAP3K14 Q99558 1/20 0.37
AKR1B1 P15121 3/20 0.35
AKR1B10 O60218 1/20 0.35
MAPT P10636 1/20 0.35
AKR1A1 P14550 1/20 0.35
BACE1 P56817 2/20 0.34
APP P05067 1/20 0.34
CYP26A1 O43174 1/20 0.33
CYP26B1 Q9NR63 1/20 0.33
OPRD1 P41143 2/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579800 0.74 CYP1A2 (0.54) MAPTKDM4EMEN1ALDH1A1KMT2A
SCHEMBL17802125 0.71 MAPT (0.46) AKR1B1AKR1B10MAPTAKR1A1BACE1
SCHEMBL11926956 0.71 BACE1 (0.42) AKR1B1AKR1B10MAPTAKR1A1BACE1
SCHEMBL15542586 0.71 MAPT (0.44) BRAFKDRAKR1B1AKR1B10MAPT
SCHEMBL16907583 0.71 ALDH1A1 (0.59) BRAFKDRMAPTKDM4EMEN1
SCHEMBL15541888 0.69 RAB9A (0.41) AKR1B1MAPTMEN1ALDH1A1KMT2A
SCHEMBL30134236 0.69 KDM4E (0.53) BRAFKDRAKR1B1MAPTCYP26A1
SCHEMBL20939584 0.68 DYRK1A (0.47) MAPTKDM4EMEN1ALDH1A1KMT2A
SCHEMBL28332239 0.68 KCNH2 (0.38) MAPTKDM4EMEN1ALDH1A1KMT2A
SCHEMBL12533417 0.68 PDK2 (0.37) BRAFKDRAKR1B1AKR1B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2864289-B1 CYCLOPROPANECARBOXAMIDO-SUBSTITUTED AROMATIC COMPOUNDS AS ANTI-TUMOR AGENTS CB THERAPEUTICS INC (KY) 2018-04-11 EP disclosed