SCHEMBL2004134

SCHEMBL2004134

CCOc1ccc2c(c1)c(C(=O)c1nc(-c3ccccn3)no1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 1/20 0.40
ALOX5AP P20292 8/20 0.40
ALOX5 P09917 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
FAAH O00519 1/20 0.38
CES1 P23141 1/20 0.38
NCEH1 Q6PIU2 1/20 0.38
DAGLA Q9Y4D2 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002804 0.94 NPC1 (0.45) SMN1; SMN2MAPTKMT2ACYP3A4CYP2C9
SCHEMBL2004994 0.93 MAPT (0.44) MAPTKMT2ACYP3A4CYP2C9LMNA
SCHEMBL2001259 0.91 SMN1; SMN2 (0.39) SMN1; SMN2MAPTKMT2AALOX5APNPC1
SCHEMBL2006770 0.90 GRM5 (0.42) SMN1; SMN2MAPTKMT2ACYP3A4NPC1
SCHEMBL2007692 0.90 ALOX5AP (0.39) SMN1; SMN2MAPTKMT2AALOX5APALOX5
SCHEMBL2004420 0.89 FAAH (0.44) SMN1; SMN2MAPTKMT2ANPC1RAB9A
SCHEMBL2003750 0.88 FAAH (0.40) SMN1; SMN2MAPTKMT2ANPC1RAB9A
SCHEMBL2005817 0.87 SMPD1 (0.44) SMN1; SMN2MAPTKMT2AALOX5APALOX5
SCHEMBL2001509 0.86 FAAH (0.43) KMT2AFAAHCES1NCEH1DAGLA
SCHEMBL2002872 0.86 PLA2G2A (0.49) SMN1; SMN2MAPTKMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed