SCHEMBL20042758

SCHEMBL20042758

CCc1nc(O)c2c(n1)CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTOR P42345 3/20 0.40
PARP1 P09874 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
C5AR1 P21730 2/20 0.36
ESR2 Q92731 1/20 0.34
USP2 O75604 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADORA1 P30542 1/20 0.34
DDB1 Q16531 2/20 0.34
CRBN Q96SW2 2/20 0.34
NR1H2 P55055 2/20 0.33
MAPT P10636 1/20 0.33
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
POLB P06746 1/20 0.33
MKNK1 Q9BUB5 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31615021 1.00 MTOR (0.40) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL31016562 0.82 C5AR1 (0.39) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL20042662 0.82 C5AR1 (0.39) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL20042672 0.82 MTOR (0.49) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL31614769 0.82 MTOR (0.49) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL31016608 0.80 PARP1 (0.37) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL20042678 0.78 DDB1 (0.39) MTORPARP1TNKS2PARP2C5AR1
SCHEMBL29329889 0.77 PARP1 (0.44) MTORPARP1TNKS2PARP2ESR2
SCHEMBL1262659 0.76 PARP1 (0.43) MTORPARP1TNKS2PARP2ESR2
SCHEMBL22503993 0.75 DDB1 (0.51) ESR2DDB1CRBNNR1H2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed