SCHEMBL20042761

SCHEMBL20042761

CC(C)(C)OC(=O)N1Cc2nc(C3CC3)nc(N3CCC3)c2C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTOR P42345 3/20 0.44
CHRM3 P20309 8/20 0.42
PDE4A P27815 6/20 0.42
PDE4B Q07343 6/20 0.42
PDE4C Q08493 6/20 0.42
PDE4D Q08499 6/20 0.42
PDE10A Q9Y233 3/20 0.40
GPR119 Q8TDV5 1/20 0.37
PDE8B O95263 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
HPGD P15428 1/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042974 0.93 MTOR (0.49) MTORCHRM3PDE4APDE4BPDE4C
SCHEMBL20042972 0.83 MTOR (0.47) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL31614795 0.83 MTOR (0.47) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL20042670 0.83 MTOR (0.47) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL31516224 0.82 MTOR (0.46) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL20042815 0.82 MTOR (0.46) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL20042678 0.82 DDB1 (0.39) MTORGPR119PDE8BDDB1CRBN
SCHEMBL20042708 0.81 MTOR (0.46) MTORPDE10AGPR119CKS1BSKP1
SCHEMBL20042676 0.81 DDB1 (0.38) MTORPDE10AGPR119PDE8BDDB1
SCHEMBL20042818 0.81 MTOR (0.46) MTORPDE10AGPR119CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed