SCHEMBL20042860

SCHEMBL20042860

CCc1nc2c(c(N3CCC3)n1)C(C)N(C(=O)c1cccc(C#N)c1)C2

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.40
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
CASR P41180 1/20 0.37
SMO Q99835 1/20 0.37
NAMPT P43490 2/20 0.36
ADORA2A P29274 5/20 0.36
GSK3B P49841 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042894 0.88 GRM5 (0.40) GRM5HCRTR1HCRTR2CASRSMO
SCHEMBL20042843 0.88 GRM5 (0.40) GRM5HCRTR1HCRTR2CASRSMO
SCHEMBL20042922 0.86 TACR2 (0.40) MEN1ALDH1A1RECQLKMT2ANPSR1
SCHEMBL20042989 0.86 SMN1; SMN2 (0.44) GRM5MEN1ALDH1A1KMT2A
SCHEMBL20042932 0.86 GRM5 (0.38) GRM5HCRTR1HCRTR2CASRSMO
SCHEMBL20042928 0.80 TACR3 (0.44) GRM5MEN1ALDH1A1RECQLKMT2A
SCHEMBL20042835 0.80 HSD17B10 (0.41) MEN1ALDH1A1RECQLKMT2ANPSR1
SCHEMBL20042767 0.76 TACR3 (0.44) GRM5ALDH1A1
SCHEMBL20042939 0.75 GRM5 (0.40) GRM5MEN1ALDH1A1KMT2A
SCHEMBL20042853 0.75 GPR6 (0.34) HCRTR1HCRTR2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed