SCHEMBL20042767

SCHEMBL20042767

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1ccc(C#N)cc1)C2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.44
KCNH2 Q12809 1/20 0.44
ALDH1A1 P00352 1/20 0.40
P2RX7 Q99572 1/20 0.39
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
PDK2 Q15119 3/20 0.38
PDK1 Q15118 2/20 0.38
PDK3 Q15120 2/20 0.38
PDK4 Q16654 2/20 0.38
GRM5 P41594 1/20 0.38
FASN P49327 7/20 0.38
DPP4 P27487 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
PDE2A O00408 1/20 0.35
SLC6A7 Q99884 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042894 0.88 GRM5 (0.40) P2RX7GRM5PDE2A
SCHEMBL20042843 0.88 GRM5 (0.40) P2RX7GRM5PDE2A
SCHEMBL20043019 0.87 POLB (0.34) TACR3KCNH2ALDH1A1P2RX7GRM5
SCHEMBL20042982 0.86 P2RX7 (0.46) TACR3KCNH2ALDH1A1P2RX7SLC6A7
SCHEMBL20042865 0.86 TACR3 (0.42) TACR3KCNH2
SCHEMBL20042851 0.86 P2RX7 (0.46) TACR3KCNH2ALDH1A1P2RX7SLC6A7
SCHEMBL20042958 0.86 TACR3 (0.42) TACR3KCNH2
SCHEMBL20042897 0.86 ALDH1A1 (0.40) ALDH1A1P2RX7FASN
SCHEMBL20042939 0.85 GRM5 (0.40) TACR3KCNH2ALDH1A1P2RX7GRM5
SCHEMBL20042853 0.85 GPR6 (0.34) TACR3KCNH2ALDH1A1P2RX7FASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed