SCHEMBL20042894

SCHEMBL20042894

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1cccc(C#N)c1)C2

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.40
CASR P41180 1/20 0.39
PDE2A O00408 2/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
P2RX7 Q99572 2/20 0.37
SMO Q99835 1/20 0.36
LRRK2 Q5S007 1/20 0.36
CNR2 P34972 1/20 0.36
GPR6 P46095 1/20 0.36
ELANE P08246 1/20 0.36
NAMPT P43490 1/20 0.35
MAP3K12 Q12852 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042843 1.00 GRM5 (0.40) GRM5CASRPDE2AHCRTR1HCRTR2
SCHEMBL20042767 0.88 TACR3 (0.44) GRM5PDE2AP2RX7
SCHEMBL20042860 0.88 GRM5 (0.40) GRM5CASRHCRTR1HCRTR2SMO
SCHEMBL20042932 0.88 GRM5 (0.38) GRM5CASRPDE2AHCRTR1HCRTR2
SCHEMBL20043019 0.88 POLB (0.34) GRM5P2RX7
SCHEMBL20042853 0.86 GPR6 (0.34) HCRTR1HCRTR2P2RX7GPR6
SCHEMBL20042939 0.86 GRM5 (0.40) GRM5P2RX7
SCHEMBL20042841 0.85 TACR2 (0.45) GRM5
SCHEMBL20042898 0.85 TACR3 (0.45) GRM5P2RX7
SCHEMBL20042897 0.85 ALDH1A1 (0.40) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed