SCHEMBL20042877

SCHEMBL20042877

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1ccc(C(F)F)c(Cl)c1)C2

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 12/20 0.36
TACR2 P21452 10/20 0.36
TACR1 P25103 8/20 0.36
KCNH2 Q12809 3/20 0.36
P2RX7 Q99572 3/20 0.34
RORC P51449 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.32
HPGD P15428 1/20 0.32
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042889 0.93 TACR3 (0.36) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042879 0.90 TACR3 (0.36) TACR3TACR2TACR1KCNH2
SCHEMBL20042852 0.88 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042914 0.87 NPSR1 (0.38) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042878 0.86 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042727 0.86 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042983 0.86 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042883 0.86 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042918 0.85 TACR3 (0.36) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042982 0.83 P2RX7 (0.46) TACR3TACR2TACR1KCNH2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed