SCHEMBL20042883

SCHEMBL20042883

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1ccc(Cl)c(C)c1)C2

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 1/20 0.39
TACR3 P29371 10/20 0.38
TACR2 P21452 8/20 0.38
TACR1 P25103 6/20 0.38
KCNH2 Q12809 3/20 0.38
LMNA P02545 1/20 0.36
P2RX7 Q99572 1/20 0.36
THRB P10828 2/20 0.35
TP53 P04637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GPR183 P32249 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042983 1.00 GPR6 (0.39) GPR6TACR3TACR2TACR1KCNH2
SCHEMBL20042878 0.90 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042727 0.90 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042852 0.88 TACR3 (0.47) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042900 0.88 TACR3 (0.38) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042889 0.88 TACR3 (0.36) TACR3TACR2TACR1KCNH2LMNA
SCHEMBL20043017 0.88 ALDH1A1 (0.36) TACR3TACR2TACR1KCNH2LMNA
SCHEMBL20042851 0.88 P2RX7 (0.46) TACR3TACR2TACR1KCNH2LMNA
SCHEMBL20042982 0.88 P2RX7 (0.46) TACR3TACR2TACR1KCNH2LMNA
SCHEMBL20042841 0.86 TACR2 (0.45) TACR3TACR2KCNH2LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed