SCHEMBL20042852

SCHEMBL20042852

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1ccc(F)c(Cl)c1)C2

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 15/20 0.47
TACR2 P21452 9/20 0.47
TACR1 P25103 7/20 0.47
KCNH2 Q12809 4/20 0.47
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
PDE2A O00408 1/20 0.37
P2RX7 Q99572 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042727 0.92 TACR3 (0.47) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042878 0.92 TACR3 (0.47) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042900 0.90 TACR3 (0.38) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042983 0.88 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042883 0.88 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042982 0.88 P2RX7 (0.46) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042851 0.88 P2RX7 (0.46) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042877 0.88 TACR3 (0.36) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042841 0.86 TACR2 (0.45) TACR3TACR2KCNH2
SCHEMBL20042753 0.86 ALDH1A1 (0.36) TACR3TACR2TACR1KCNH2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed