SCHEMBL20042881

SCHEMBL20042881

C1CN(c2nc3c(c(N4CCC4)n2)CNC3)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.41
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR2C P28335 2/20 0.40
HTR2A P28223 1/20 0.39
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
CASP1 P29466 1/20 0.36
CASP4 P49662 1/20 0.36
CASP5 P51878 1/20 0.36
GLA P06280 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042683 0.81 NPY5R (0.39) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL20042813 0.81 HTR2C (0.37) SMN1; SMN2HTR2CPDE4APDE4BPDE4C
SCHEMBL31614818 0.81 NPY5R (0.39) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL20042777 0.81 HRH4 (0.38) HRH1HTR2CHTR2A
Hydrochloric Acid SCHEMBL31405518 0.79 MEN1 (0.39) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL31614730 0.79 MEN1 (0.39) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL19358098 0.77 HRH4 (0.41)
SCHEMBL20042692 0.77 MTOR (0.37) USP2HTR2CHTR2ATSHRHSD17B10
SCHEMBL31615106 0.77 MTOR (0.37) USP2HTR2CHTR2ATSHRHSD17B10
SCHEMBL20042648 0.77 CHRM3 (0.51) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed