SCHEMBL20042777

SCHEMBL20042777

Nc1nc2c(c(N3CCC3)n1)CNC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 15/20 0.38
CHUK O15111 1/20 0.38
LMNA P02545 1/20 0.37
HRH3 Q9Y5N1 2/20 0.35
ADRB1 P08588 1/20 0.34
TACR2 P21452 1/20 0.34
ADRA1D P25100 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
CCR1 P32246 1/20 0.34
HRH1 P35367 1/20 0.34
AVPR1A P37288 1/20 0.34
HTR2B P41595 1/20 0.34
HTR3A P46098 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
NPY5R Q15761 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19358098 0.97 HRH4 (0.41) HRH4CHUKLMNAHRH3NPY5R
Trifluoroacetic Acid SCHEMBL29710241 0.83 LMNA (0.35) HRH4CHUKLMNAHRH3NPY5R
SCHEMBL20042881 0.81 HRH1 (0.41) HTR2AHTR2CHRH1
SCHEMBL20042813 0.79 HTR2C (0.37) HTR2C
SCHEMBL20042683 0.79 NPY5R (0.39) NPY5R
SCHEMBL31614818 0.79 NPY5R (0.39) NPY5R
Hydrochloric Acid SCHEMBL31614730 0.78 MEN1 (0.39) NPY5R
Hydrochloric Acid SCHEMBL31405518 0.78 MEN1 (0.39) NPY5R
SCHEMBL20042692 0.76 MTOR (0.37) HRH4LMNAHTR2AHTR2CHTR2B
SCHEMBL31615106 0.76 MTOR (0.37) HRH4LMNAHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed