SCHEMBL2004561

SCHEMBL2004561

O=C(c1noc(-c2cccnc2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(O)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 4/20 0.38
L3MBTL1 Q9Y468 3/20 0.36
S1PR1 P21453 1/20 0.34
LMNA P02545 4/20 0.34
MAPT P10636 4/20 0.34
ALDH1A1 P00352 3/20 0.34
ALOX12 P18054 2/20 0.34
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
KDM4E B2RXH2 2/20 0.33
EPHX2 P34913 1/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 3/20 0.33
TSHR P16473 1/20 0.33
CHRNB2 P17787 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004314 0.95 RET (0.39) RETL3MBTL1S1PR1LMNAMAPT
SCHEMBL2002558 0.92 RET (0.39) RETL3MBTL1S1PR1LMNAMAPT
SCHEMBL2005007 0.92 PTGES2 (0.40) RETS1PR1MAPTALDH1A1ALOX12
SCHEMBL2000706 0.92 RET (0.39) RETL3MBTL1S1PR1LMNAMAPT
SCHEMBL2003892 0.91 L3MBTL1 (0.36) RETL3MBTL1LMNAMAPTALDH1A1
SCHEMBL2006526 0.90 L3MBTL1 (0.39) RETL3MBTL1LMNAMAPTALDH1A1
SCHEMBL2010388 0.90 MAPT (0.39) RETL3MBTL1LMNAMAPTCYP17A1
SCHEMBL2007600 0.89 S1PR1 (0.40) RETL3MBTL1S1PR1LMNAMAPT
SCHEMBL2004983 0.88 PTGES2 (0.42) RETS1PR1MAPTALDH1A1ALOX12
SCHEMBL2000312 0.87 LMNA (0.39) RETL3MBTL1LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed