SCHEMBL2010388

SCHEMBL2010388

COc1ccc2c(c1)c(C(=O)c1noc(-c3cccnc3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
TP53 P04637 5/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
DGAT2 Q96PD7 1/20 0.38
RET P07949 3/20 0.38
PLA2G2A P14555 2/20 0.37
CYP17A1 P05093 2/20 0.37
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007600 0.93 S1PR1 (0.40) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL2004314 0.93 RET (0.39) MAPTNPC1RAB9ARETPKM
SCHEMBL2002012 0.92 PTGES2 (0.40) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL2001214 0.91 PLA2G2A (0.38) MAPTTP53NPC1RAB9ACYP3A4
SCHEMBL2002558 0.91 RET (0.39) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL2002749 0.91 NPC1 (0.41) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL2004561 0.90 RET (0.38) MAPTNPC1RAB9ACYP3A4RET
SCHEMBL2000706 0.89 RET (0.39) MAPTTP53SMN1; SMN2CYP3A4CYP1A2
SCHEMBL2002120 0.89 ABCB1 (0.41) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL2004484 0.88 KDM4E (0.38) MAPTTP53NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed