SCHEMBL20049948

SCHEMBL20049948

C=C(C)Nc1ncc(-c2cc(C(F)(F)F)ccc2C)cc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2B Q13224 3/20 0.43
KDR P35968 7/20 0.40
MAPK14 Q16539 6/20 0.40
LCK P06239 6/20 0.40
JAK3 P52333 5/20 0.40
TEK Q02763 3/20 0.40
NOTUM Q6P988 1/20 0.36
DDR2 Q16832 1/20 0.36
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BRAF P15056 4/20 0.36
RAF1 P04049 3/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20049967 0.82 ALDH1A1 (0.52) GRIN1GRIN2BALDH1A1L3MBTL1SLC1A3
SCHEMBL20049992 0.79 CNR1 (0.39) ABL1GRIN1GRIN2BKDRMAPK14
SCHEMBL20049904 0.76 GRIN2B (0.42) ABL1GRIN1GRIN2BALDH1A1
SCHEMBL25588581 0.76 EPHB4 (0.42) TEKTRPV1
SCHEMBL20049825 0.73 GSK3B (0.42) GRIN1GRIN2BALDH1A1MAPK13MAPK12
SCHEMBL20050027 0.73 GRIN2B (0.44) GRIN1GRIN2B
SCHEMBL20049775 0.73 NPC1 (0.42) ABL1GRIN1GRIN2BKDRTEK
SCHEMBL20049886 0.73 PSMB5 (0.42) KDR
SCHEMBL25588074 0.73 CHRNA7 (0.38) ALDH1A1L3MBTL1
SCHEMBL25584752 0.72 GRIN2B (0.43) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067786-A1 SUBSTITUTED 1H-IMIDAZO[4,5-B]PYRIDIN-2(3H)-ONES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-04-12 WO disclosed