SCHEMBL2004999

SCHEMBL2004999

CCOc1ccc2c(c1)c(C(=O)c1nnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 10/20 0.40
ALOX5 P09917 5/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
OPRK1 P41145 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004726 0.94 OPRK1 (0.42) ALOX5APALOX5CYP3A4CYP2C9OPRK1
SCHEMBL2004340 0.91 F2RL3 (0.37) ALOX5APOPRK1MAPTSMN1; SMN2
SCHEMBL2004657 0.91 FAAH (0.38) ALOX5APALOX5CYP3A4CYP2C9OPRK1
SCHEMBL2003878 0.90 ALOX5AP (0.39) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL2004616 0.90 ALOX5AP (0.42) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL2008229 0.90 ALOX5AP (0.40) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL1999807 0.89 ALOX5AP (0.42) ALOX5APALOX5CYP3A4CYP2C9PTGS1
SCHEMBL2002574 0.89 FAAH (0.42) OPRK1MAPTKMT2A
SCHEMBL2002177 0.88 MAPT (0.38) ALOX5APALOX5CYP3A4CYP2C9OPRK1
SCHEMBL2008081 0.88 FAAH (0.41) ALOX5APALOX5CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed