SCHEMBL20050000

SCHEMBL20050000

C=C(C)Nc1ncc(-c2cc(F)ccc2CCC)cc1C

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 9/20 0.39
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CHRNA7 P36544 1/20 0.35
GRIN1 Q05586 3/20 0.35
GRIN2B Q13224 3/20 0.35
GCGR P47871 1/20 0.33
NR3C2 P08235 1/20 0.33
RAB9A P51151 1/20 0.33
F2RL1 P55085 2/20 0.32
CASP6 P55212 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25588082 0.84 CHRNA7 (0.39) ABL1CHRNA7GRIN1GRIN2BF2RL1
SCHEMBL20049904 0.81 GRIN2B (0.42) ABL1NPC1ALDH1A1GRIN1GRIN2B
SCHEMBL20049775 0.79 NPC1 (0.42) ABL1NPC1ALDH1A1CHRNA7GRIN1
SCHEMBL20049838 0.74 NPC1 (0.38) ABL1NPC1ALDH1A1GRIN1GRIN2B
SCHEMBL20050025 0.74 CDK8 (0.39) GRIN1GRIN2B
SCHEMBL20049970 0.74 GRM5 (0.43) NPC1ALDH1A1GRIN1GRIN2BRAB9A
SCHEMBL20049825 0.73 GSK3B (0.42) NPC1ALDH1A1GRIN1GRIN2B
SCHEMBL20050027 0.73 GRIN2B (0.44) GRIN1GRIN2B
SCHEMBL20049992 0.73 CNR1 (0.39) ABL1NPC1ALDH1A1GRIN1GRIN2B
SCHEMBL25587881 0.72 ABL1 (0.44) ABL1NPC1ALDH1A1CHRNA7GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067786-A1 SUBSTITUTED 1H-IMIDAZO[4,5-B]PYRIDIN-2(3H)-ONES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-04-12 WO disclosed