SCHEMBL20050146

SCHEMBL20050146

C=C/C=C\C=C(/C)C(CNCC(O)COc1ccc(C2CCCCC2)cc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.41
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
LMNA P02545 2/20 0.40
HTR1A P08908 1/20 0.37
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
CYP2D6 P10635 1/20 0.36
ADRB3 P13945 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20049943 0.80 MEN1 (0.56) ABCB1KMT2AMEN1OPRM1OPRD1
SCHEMBL20049942 0.74 ADRB2 (0.51) KMT2AMEN1OPRM1OPRD1LMNA
SCHEMBL8681927 0.67 MEN1 (0.49) KMT2AMEN1CYP2D6
SCHEMBL24433964 0.66 ADRB2 (0.40) KMT2AMEN1OPRM1OPRD1LMNA
SCHEMBL1803614 0.64 LMNA (0.51) KMT2AMEN1LMNA
SCHEMBL11606524 0.64 MEN1 (0.71) KMT2AMEN1OPRM1OPRD1LMNA
SCHEMBL20049936 0.63 POLB (0.57) KMT2AMEN1LMNACYP2D6
SCHEMBL18965637 0.63 LMNA (0.44) KMT2AMEN1LMNAADRB2ADRB1
SCHEMBL28000803 0.63 LMNA (0.53) KMT2AMEN1LMNA
SCHEMBL20049939 0.63 MEN1 (0.75) ABCB1KMT2AMEN1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067685-A1 SMALL MOLECULE AMPK ACTIVATORS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2018-04-12 WO disclosed