SCHEMBL20051946

SCHEMBL20051946

NN1CCC2(CC1)CCN(CC(F)F)CC2

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 11/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25001373 0.79 CYP2D6 (0.41) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL18497937 0.78 TSHR (0.46) CYP2D6SMN1; SMN2CYP2C9TSHRALDH1A1
SCHEMBL18517451 0.75 TSHR (0.38) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL24940878 0.73 CYP2D6 (0.37) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL23126657 0.71 MAPT (0.49) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL18517454 0.71 TSHR (0.50) CYP2D6CYP2C9TSHRALDH1A1CYP3A4
SCHEMBL29326370 0.68 CYP2D6 (0.38) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL18517455 0.68 CYP2D6 (0.43) CYP2D6OPRM1OPRD1OPRK1CYP2C9
SCHEMBL23514830 0.68 OPRM1 (0.39) CYP2D6SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL18517453 0.68 TSHR (0.43) CYP2D6CYP2C9TSHRALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944613-B2 Fumagillol spirocyclic compounds and fused bicyclic compounds and methods of making and using same ZAFGEN, INC. (US) 2018-04-17 US disclosed
US-9944613-B2 Fumagillol spirocyclic compounds and fused bicyclic compounds and methods of making and using same ZAFGEN, INC. (US) 2018-04-17 US disclosed