SCHEMBL20052420

SCHEMBL20052420

CC(C)[C@H](NC(=O)C(Cc1cn(C)c2ccccc12)NC(=O)C(CC(=O)OC(C)(C)C)NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 6/20 0.47
CASP7 P55210 3/20 0.45
CASP1 P29466 3/20 0.45
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
IDO1 P14902 2/20 0.43
ECE1 P42892 2/20 0.42
MME P08473 1/20 0.42
REN P00797 2/20 0.42
CTSB P07858 2/20 0.41
CTSK P43235 1/20 0.41
CTSL P07711 1/20 0.41
NMBR P28336 1/20 0.41
CASP9 P55211 2/20 0.40
CCKAR P32238 1/20 0.40
CCKBR P32239 1/20 0.40
OPRD1 P41143 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20052423 1.00 CASP3 (0.47) CASP3CASP7CASP1MMP9MMP8
SCHEMBL20052446 0.92 CASP3 (0.43) CASP3CASP7CASP1ECE1MME
SCHEMBL20356041 0.92 CASP3 (0.43) CASP3CASP7CASP1ECE1MME
SCHEMBL19944793 0.91 CASP3 (0.45) CASP3CASP7CASP1MMP9MMP8
SCHEMBL20052454 0.91 CASP3 (0.45) CASP3CASP7CASP1MMP9MMP8
SCHEMBL15462692 0.89 MMP9 (0.46) CASP3MMP9MMP8IDO1REN
SCHEMBL15462695 0.87 CASP3 (0.65) CASP3CASP7CASP1CASP9
SCHEMBL20355913 0.87 CASP3 (0.65) CASP3CASP7CASP1CASP9
SCHEMBL20355912 0.87 CASP3 (0.65) CASP3CASP7CASP1CASP9
SCHEMBL20052371 0.87 CASP3 (0.65) CASP3CASP7CASP1CASP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944674-B2 Selective cysteine protease inhibitors and uses thereof GENESIS TECHNOLOGIES LIMITED (BB) 2018-04-17 US disclosed