SCHEMBL20052446

SCHEMBL20052446

CC(C)[C@H](NC(=O)[C@H](CCc1cn(C)c2ccccc12)NC(=O)C(CC(=O)OC(C)(C)C)NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 8/20 0.43
CASP1 P29466 4/20 0.43
CASP7 P55210 4/20 0.43
CASP9 P55211 3/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CTSL P07711 1/20 0.41
CTSK P43235 4/20 0.40
CTSB P07858 1/20 0.40
ECE1 P42892 2/20 0.40
MME P08473 1/20 0.40
CASP4 P49662 1/20 0.39
CASP8 Q14790 1/20 0.39
CASP10 Q92851 1/20 0.39
PSMB5 P28074 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20356041 1.00 CASP3 (0.43) CASP3CASP1CASP7CASP9MEN1
SCHEMBL20052420 0.92 CASP3 (0.47) CASP3CASP1CASP7CASP9CTSL
SCHEMBL20052423 0.92 CASP3 (0.47) CASP3CASP1CASP7CASP9CTSL
SCHEMBL20356118 0.91 CASP3 (0.42) CASP3CASP1CASP7CASP9MEN1
SCHEMBL20052427 0.87 CASP3 (0.61) CASP3CASP1CASP7CASP9CASP4
SCHEMBL7886933 0.84 CTSK (0.53) CASP3CASP1CASP7CASP9CTSL
SCHEMBL20052454 0.83 CASP3 (0.45) CASP3CASP1CASP7CASP9CTSL
SCHEMBL19944793 0.83 CASP3 (0.45) CASP3CASP1CASP7CASP9CTSL
SCHEMBL20740990 0.83 CASP3 (0.54) CASP3CASP1CASP7CASP9CTSL
SCHEMBL19015971 0.83 CASP3 (0.54) CASP3CASP1CASP7CASP9CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944674-B2 Selective cysteine protease inhibitors and uses thereof GENESIS TECHNOLOGIES LIMITED (BB) 2018-04-17 US disclosed